Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign

Linciano, Cullia, Borsari, Santucci, Ferrari, Witt, Gul, Kuzikov, Ellinger, Santarém, Cordeiro da Silva, Conti, Bolognesi, Roberti, Prati, Bartoccini, Retini, Piersanti, Cavalli, Goldoni, Bertozzi, Bertozzi, Brambilla, Rizzo, Piomelli, Pinto, Bandiera, Costi (2020) Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign Eur J Med Chem (IF: 6.7) 189 112047

Links

http://www.ncbi.nlm.nih.gov/pubmed/31982652
http://dx.doi.org/10.1016/j.ejmech.2020.112047

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